BTRX335140 Datasheet DC Chemicals
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Cat.No DC23413
Name BTRX335140

Chemical Properties

CAS 2244614-14-8
Formula C25H32FN5O2
MW 453.552289009094
Storage 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Biological activity

Description CAS NO.：2244614-14-8
Product Name：BTRX-335140
Synonyms：XK5ILZ28KI;GTPL10452;BTRX335140;CYM53093;compound 58 [PMID: 30707578];4-Piperidinamine, 1-(6-ethyl-8-fluoro-4-methyl-3-(3-methyl-1,2,4-oxadiazol-5-yl)-2-quinolinyl)-N-(tetrahydro-2H-pyran-4-yl)-;1-[6-ethyl-8-fluoro-4-methyl-3-(3-methyl-1,2,4-oxadiazol-5-yl)quinolin-2-yl]-N-(oxan-4-yl)piperidin-4-amine;1-(6-Ethyl-8-fluoro-4-methyl-3-(3-methyl-1,2,4-oxadiazol-5-yl)quinolin-2-yl)-N-(tetrahydro-2H-pyran-4-yl)pipe;Unii-XK5ilz28KI;BTRX-335140;Navacaprant
EINEC:
Molecular Formula：C25H32FN5O2
Molecular Weight：453.552289009094
Target: IC50: 0.8 nM (κOR); 110 nM (μOR); 6500 nM (δOR)[1]
In Vivo
In Vitro
Kinase Assay
Cell Assay
Animal Administration

References

[1]. Guerrero M, et al. Design and Synthesis of a Novel and Selective Kappa Opioid Receptor (KOR) Antagonist (BTRX-335140). J Med Chem. 2019 Feb 28;62(4):1761-1780.
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