TAN-452 Datasheet DC Chemicals

Description	TAN-452 is an orally active, selective peripherally acting δ-opioid receptor (DOR) antagonist with a Ki of 0.47?nM and a Kb of 0.21?nM. TAN-452 is an antagonist for μ-opioid receptor (MOR; Ki=36.56?nM and Kb=9.43?nM) and κ-opioid receptor (KOR; Ki=5.31?nM and Kb=7.18?nM). TAN-452, a derivative of Naltrindole, demonstrates low brain penetrability and attenuates morphine-induced side effects without affecting pain control.
Cat.No	DC40852
Name	TAN-452

Chemical Properties

CAS	892039-23-5
Formula	C29H30N2O5
MW	486.56
Storage	Please store the product under the recommended conditions in the Certificate of Analysis.

References

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