Chemical Properties
CAS |
13187-06-9 |
|
Formula |
C23H23NO4S |
MW |
409.498025178909 |
Storage |
2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO |
Biological activity
Description |
CAS NO.:13187-06-9 Product Name:9-(1-Methyl-4-piperidylene)thioxanthene maleate Synonyms:9-(1-Methyl-4-piperidylene)thioxanthene maleate;1-METHYL-4-[THIOXANTHEN-9-YLIDENE]PIPERIDINE MALEATE SALT;PIMETHIXEN MALEATE SALT;Pimethixene maleate salt;1-methyl-4-(9H-thioxanthen-9-ylidene)piperidinium hydrogen maleate;1-Methyl-4-(thioxanthen-9-ylidene)piperidine;9-(1-methyl-4-piperidylene)-thioxanthenmaleate;9-(n-methyl-piperidyliden-4)thioxanemaleate;bp-400;PIMETHIXENE MALEATE;Pimethixene maleic salt;PIMETHIXENE MALEATE SALT;9-(1-methyl-4-piperidylene)thioxanthenemaleate EINEC: Molecular Formula:C23H23NO4S Molecular Weight:409.498025178909 |
Target: |
pKi: 7.63 (5-HT1A receptor), 10.22 (5-HT2A receptor), 10.44 (5-HT2B receptor), 8.42 (5-HT2C receptor), 10.14 (histamine H1 receptor), 8.19 (D2 receptor), 7.54 (DD4.4 receptor), 8.61 (M1 receptor), 9.38 (M2 receptor)[1] |
In Vivo |
|
In Vitro |
|
Kinase Assay |
|
Cell Assay |
|
Animal Administration |
|
References
[1]. Schmitz B, et al. BF-1--a novel selective 5-HT2B receptor antagonist blocking neurogenic dural plasma protein extravasation in guinea pigs. Eur J Pharmacol. 2015 Mar 15;751:73-80. |
|
Return Policy
If you are in any way unsatisfied with your purchase, you may return any item(s) within 365 days of its original purchase date.
Please provide your Order Number in the email. We strive to reply to all email inquiries within one business day.
Tel: +86-21-58447131
Fax: +86-21-61642470
Email:
sales@dcchemicals.com
order@dcchemicals.com
Website:
www.dcchemicals.com
|