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(2S,3R)-LP99

  Cat. No.:  DC71320  
Chemical Structure
1808948-28-8
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More than 5000 active chemicals with high quality for research!
Field of application
(2S,3R)-LP99 is a potent and selective BRD7 and BRD9 inhibitor with an KD of 99 nM for BRD9. (2S,3R)-LP99 inhibits the association of BRD7 and BRD9 to acetylated histones in vitro and in cells. (2S,3R)-LP99 demonstrates that BRD7/9 plays a role in regulating pro-inflammatory cytokine secretion.
Chemicals PropertiesBiological activity Related products COA MSDS Datasheet
Cas No.: 1808948-28-8
SMILES: CC(CS(=O)(N[C@@H]([C@@H](N1C2=CC3=C(C(C)=CC(N3C)=O)C=C2)C4=CC=C(C=C4)Cl)CCC1=O)=O)C
M.Wt: 516.05
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
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