BRD2492 |CAS 1821669-43-5|DC Chemicals

Cas No.:	1821669-43-5
Chemical Name:	4-Acetylamino-N-(2-amino-5-pyridin-4-yl-phenyl)-benzamide
Synonyms:	BRD2492;4-Acetylamino-N-(2-amino-5-pyridin-4-yl-phenyl)-benzamide;BDBM178095
SMILES:	O=C(C1C=CC(=CC=1)NC(C)=O)NC1C(=CC=C(C2C=CN=CC=2)C=1)N
Formula:	C₂₀H₁₈N₄O₂
M.Wt:	346.382524013519
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

BRD2492 is a highly potent, selective HDAC1/2 inhibitor (IC50=2/19 nM, respectively) that displays excellent selectivity versus HDAC3 (IC50=2.08 uM, ≥110-fold selectivity) and all other HDAC isoforms, increases caspase-3 activation.

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