Ganaplacide|KAF156|cas 1261113-96-5|DC Chemicals

Cas No.:	1261113-96-5
Chemical Name:	2-amino-1-[3-(4-fluoroanilino)-2-(4-fluorophenyl)-8,8-dimethyl-5,6-dihydroimidazo[1,2-a]pyrazin-7(8H)-yl]ethan-1-one
Synonyms:	KAF156;GNF-156
SMILES:	NCC(N1CCN2C(=C(N=C2C1(C)C)C1=CC=C(F)C=C1)NC1=CC=C(F)C=C1)=O
Formula:	C₂₂H₂₃F₂N₅O
M.Wt:	411.457
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

Ganaplacide (KAF156, GNF-156) is a novel antimalarial clinical candidate that shows blood schizonticidal activity with IC50 of 6-17.4 nM against P falciparum drug-sensitive and drug-resistant strains.

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