VX-984cas 1562396-65-9|DC Chemicals

Cas No.:	1562396-65-9
Chemical Name:	VX-984 analog
Synonyms:	BCP29319;VX-984 analog
SMILES:	O=C(C1C([H])=C([H])N=C2C=1C([H])=C([H])C([H])=C2[C@]([H])(C([H])([H])[H])C([H])([H])N([H])C1C([H])=C(C2=C([2H])N=C(C([H])([H])[H])N=C2[2H])N=C([H])N=1)N([H])[H]
Formula:	C₂₂H₂₁N₇O
M.Wt:	401.4608
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

VX-984 (M 9831) is a potent, selective inhibitor of DNA-PK with IC50 of 88±64 nM for inhibition of DNA-PKcs autophosphorylation (Ser2056) in A549 lung cancer cells, with good selectivity versus other PI3K family members.Solid TumorsPhase 1 Clinical

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