ML 278|CAS 1604821-43-3|DC Chemicals

Cas No.:	1604821-43-3
Chemical Name:	3,5-dimethoxy-N-(4-(1-(2-methoxyacetyl)indolin-5-yl)thiazol-2-yl)benzamide
Synonyms:	ML278
Formula:	C₂₃H₂₃N₃O₅S
M.Wt:	453.513
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

ML278 is a potent and reversible inhibitor of lipid uptake via SR-BI (scavenger receptor BI) with IC50 of 6 nM; a plasma-stable, noncytotoxic probe that exhibits moderate metabolic stability, thus displaying improved properties for in vitro and in vivo studies; increases the binding of HDL to SR-BI.

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