MS0124|MS 0124

Cas No.:	1197196-63-6
Chemical Name:	6,7-Dimethoxy-N-(1-Methylpiperidin-4-Yl)-2-(Morpholin-4-Yl)quinazolin-4-Amine
Synonyms:	MS0124;6,7-dimethoxy-N-(1-methylpiperidin-4-yl)-2-morpholinoquinazolin-4-amine;6,7-Dimethoxy-N-(1-Methylpiperidin-4-Yl)-2-(Morpholin-4-Yl)quinazolin-4-Amine;7L6;BDBM50300032
SMILES:	O1CCN(CC1)C1=NC2C=C(C(=CC=2C(=N1)NC1CCN(C)CC1)OC)OC
Formula:	C₂₀H₂₉N₅O₃
M.Wt:	387.475964307785
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

MS-0124 is a potent and selective inhibitor of G9a-like Protein (GLP) lysine methyltransferase with IC50 of 13 nM, shows >30-fold selectivity for GLP over G9a and other methyltransferases.

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