NVP-2|;CDK9 inhibitor|CAS 1263373-43-8|DC Chemicals

Cas No.:	1263373-43-8
Chemical Name:	4-(((2'-chloro-5'-(((1R,4r)-4-(((R)-1-methoxypropan-2-yl)amino)cyclohexyl)amino)-[2,3'-bipyridin]-6-yl)amino)methyl)tetrahydro-2H-pyran-4-carbonitrile
Synonyms:	NVP2;NVP 2;CDK9 inhibitor
SMILES:	C[C@H](COC)NC1CCC(CC1)NC2=NC=C(C(=C2)C3=NC(=CC=C3)NCC4(CCOCC4)C#N)Cl
Formula:	C₂₇H₃₇ClN₆O₂
M.Wt:	513.083
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:	NVP-2 is a CDK9 inhibitor with an IC50 of 0.5 nM.
Target:	CDK9:0.5 nM (IC50)
References:	[1]. Wang J, et al. SnapShot: Kinase Inhibitors I. Mol Cell. 2015 May 21;58(4):708.e1.

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