BI 167107|BI167107|CAS 1202235-68-4|DC Chemicals

Cas No.:	1202235-68-4
Chemical Name:	5-hydroxy-8-(1-hydroxy-2-((2-methyl-1-(o-tolyl)propan-2-yl)amino)ethyl)-2H-benzo[b][1,4]oxazin-3(4H)-one
Synonyms:	BI 167107\|BI167107
SMILES:	CC(NCC(C1C2OCC(=O)NC=2C(O)=CC=1)O)(C)CC1C=CC=CC=1C
Formula:	C₂₁H₂₆N₂O₄
M.Wt:	370.449
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Publication:	[1]. Rasmussen SG, et al. Structure of a nanobody-stabilized active state of the β(2) adrenoceptor. Nature. 2011 Jan 13;469(7329):175-80.

Description:	BI-167107 is a high affinity, full agonist that binds to the β2 adrenergic receptor (β2AR) with a dissociation constant Kd of 84 pM[1].
Target:	Kd: 84 pM (β2AR)[1]
References:	[1]. Rasmussen SG, et al. Structure of a nanobody-stabilized active state of the β(2) adrenoceptor. Nature. 2011 Jan 13;469(7329):175-80.

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