HOIPIN-1|JTP-0819958;HOIP inhibitor-1|DC Chemicals

Cas No.:
Chemical Name:	Sodium (E)-2-(3-(2-methoxyphenyl)-3-oxoprop-1-en-1-yl)benzoate
Synonyms:	HOIPIN-1\|JTP-0819958;HOIP inhibitor-1
Formula:	C₁₇H₁₃NaO₄
M.Wt:	304.277
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

HOIPIN-1 (JTP-0819958, HOIP inhibitor-1) is a chemical inhibitor of linear ubiquitin chain assembly complex (LUBAC, IC50=2.8 uM), specifically generates Met1-linked linear ubiquitin chains through the ubiquitin ligase activity in HOIP, and activates the NF-kB pathway.

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HOIPIN-1(JTP-0819958;HOIP inhibitor-1)