MMV-667492| CAS 380877-02-1

Cas No.:	380877-02-1
Chemical Name:	N-[3-(Cyclohexylamino)-1,4-dioxonaphthalen-2-yl]-N-methylnitrous amide
Synonyms:	N-(3-(Cyclohexylamino)-1,4-dioxo-1,4-dihydronaphthalen-2-yl)-N-methylnitrousamide;MMV667492;NSC766733;STK529340;N-[3-(cyclohexylamino)-1,4-dioxonaphthalen-2-yl]-N-methylnitrous amide;2-(cyclohexylamino)-3-[methyl(nitroso)amino]naphthalene-1,4-dione
SMILES:	O=C1C2C=CC=CC=2C(C(=C1NC1CCCCC1)N(C)N=O)=O
Formula:	C₁₇H₁₉N₃O₃
M.Wt:	313.351063966751
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

MMV-667492 (MMV 667492, MMV667492) is a novel potent Ezrin inhibitor with Kd of 29.4 nM; exhibits potent anti-ezrin activity in all biologic assays and has better physicochemical properties for drug-likeness than NSC305787; a novel antimetastatic agent for the treatment of metastatic osteosarcoma.

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