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LY451395

  Cat. No.:  DC24030   Featured
Chemical Structure
375345-95-2
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More than 5000 active chemicals with high quality for research!
Field of application
A potent, selective, and centrally active positive allosteric modulator of AMPAR-mediated neurotransmission, which increase ion channel flux in the presence of agonist by suppressing desensitization and/or deactivation of the receptors..
Cas No.: 375345-95-2
Chemical Name: Mibampator
Synonyms: MIBAMPATOR;N-[(2R)-2-[4-[4-[2-(methanesulfonamido)ethyl]phenyl]phenyl]propyl]propane-2-sulfonamide;{(2R)-2-[4-(4-{2-[(methylsulfonyl)amino]ethyl}phenyl)phenyl]propyl}[(methylet;2-Propanesulfonamide, N-((2R)-2-(4'-(2-((methylsulfonyl)amino)ethyl)(1,1'-biphenyl)-4-yl)propyl)-;2-PROPANESULFONAMIDE, N-[(2R)-2-[4'-[2-[(METHYLSULFONYL)AMINO]ETHYL][1,1'-BIPHENYL]-4-YL]PROPYL]-;CHEMBL1277001;CTK4H8360;LY 451395;LY-451395;Mibampator [USAN:INN];N-[(2R)-2-[4'-[2-[(Methylsulfonyl)amino]ethyl][1,1'-biphenyl]-4-yl]propyl];UNII-A9V5BW73UU;[(2R)-2-[4-[4-[2-[(Methylsulfonyl)amino]ethyl]phenyl]phenyl]propyl][(1-methylethyl)sulfonyl]amine;LY451395;AKOS027338712;MIBAMPATOR [WHO-DD];(R)-N-(2-(4'-(2-(Methylsulfonamido)ethyl)-[1,1'-biphenyl]-4-yl)propyl)propane-2-sulfonamide;BDBM50330415;LY-451395; LY451395; Mibampator;NS00068333;NCGC00390642-01;Mibampator (USAN/INN);375345-95-2;CS-3166;A9V5BW73UU;((2R)-2-(4-(4-(2-((METHYLSULFONYL)AMINO)ETHYL)PHENYL)PHENYL)PROPYL)((1-METHYLETHYL)SULFONYL)AMINE;N-[(2R)-2-[4-[4-[2-(methylsulfonylamino)ethyl]phenyl]phenyl]propyl]propane-2-sulfonamide;BCP28335;HY-10934;(R)-N-(2-(4''-(2-(methylsulfonamido)ethyl)biphenyl-4-yl)propyl)propane-2-sulfonamide;D09931;SCHEMBL3045499;DB12717;MS-27869;DA-55465;DTXSID20190977;N-((2R)-2-(4'-(2-((Methylsulfonyl)amino)ethyl)biphenyl-4-yl)propyl)propane-2-sulfonamide;BRD-K42981054-001-01-9;8SO;MFCD18251566;MIBAMPATOR [USAN];MIBAMPATOR [INN];Q27273819
SMILES: C[C@@H](CNS(C(C)C)(=O)=O)C1=CC=C(C2=CC=C(CCNS(C)(=O)=O)C=C2)C=C1
Formula: C21H30N2O4S2
M.Wt: 438.6039
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: A potent, selective, and centrally active positive allosteric modulator of AMPAR-mediated neurotransmission, which increase ion channel flux in the presence of agonist by suppressing desensitization and/or deactivation of the receptors.
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