MRS1754|A2B receptor antagonist|CAS 264622-58-4|DC Chemicals

Cas No.:	264622-58-4
Chemical Name:	MRS1754,MRS-1754,MRS 1754
Synonyms:	MRS1754,MRS-1754,MRS 1754
SMILES:	CCCN1C2=C(NC(=N2)C2=CC=C(OCC(=O)NC3=CC=C(C=C3)C#N)C=C2)C(=O)N(CCC)C1=O
Formula:	C₂₆H₂₆N₆O₄
M.Wt:	486.52
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:	MRS 1754 is a selective antagonist radioligand for A2B adenosine receptor with very low affinity for A1 and A3 receptors of both humans and rats[1].
In Vitro:	The most potent displacer of [3H]MRS 1754 binding is MRS 1754. The Ki value for displacement of [3H]MRS 1754 binding to human A2B receptors expressed in HEK-293 cell membranes is 1.45±0.21 nM[1].

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