TLX agonist 1 | TLX Modulator | CAS 958323-31-4|DC Chemicals

Cas No.:	958323-31-4
Chemical Name:	CCRP2
SMILES:	O=C(N1CCN(C(C2C=CC=CC=2)C2C=CC=CC=2)CC1)C1C=C(C)N(C)N=1
Formula:	C₂₃H₂₆N₄O
M.Wt:	374.488
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Publication:	[1]. Benod C, et al. The human orphan nuclear receptor tailless (TLX, NR2E1) is druggable. PLoS One. 2014 Jun 17;9(6):e99440.

Description:	TLX agonist 1 (ccrp2) is an orphan nuclear receptor tailless (TLX, NR2E1) modulator (EC50=1μM; Kd= 650 nM). TLX agonist 1 potentiates TLX transcriptional repressive activity[1].
References:	[1]. Benod C, et al. The human orphan nuclear receptor tailless (TLX, NR2E1) is druggable. PLoS One. 2014 Jun 17;9(6):e99440.

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