Denifanstat (TVB-2640) |CAS 1399177-37-7|DC Chemicals

Cas No.:	1399177-37-7
Chemical Name:	4-(1-(4-Cyclobutyl-2-methyl-5-(5-methyl-4H-1,2,4-triazol-3- yl)benzoyl)piperidin-4-yl)benzonitrile
Synonyms:	TVB-2640,TVB 2640,TVB2640
SMILES:	C(C1C=CC(C2CCN(C(C3C(C)=CC(C4CCC4)=C(C4=NN=C(C)N4)C=3)=O)CC2)=CC=1)#N
Formula:	C₂₇H₂₉N₅O
M.Wt:	439.55
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO

Description:

TVB-2640(FASN-IN-2) is a Fatty Acid Synthase (FASN) inhibitor extracted from patent WO2012122391A1, compound 152, has an IC50 of 0.052 μM and an EC50 of 0.072 μM[1].

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