MLEB-22043|CAS |DC Chemicals

Cas No.:
Chemical Name:	MLEB-22043
SMILES:	NC1=NC(/C(C(N[C@]2([H])C(N(S(=O)(O)=O)[C@]2(C)[H])=O)=O)=N/OC(C)(C)C(NCC3=CN(CC(C(C=C(O)C(O)=C4)=C4O5)=CC5=O)N=N3)=O)=CS1
Formula:	C₂₆H₂₇N₉O₁₁S₂
M.Wt:	705.68
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Cat. No.	Product name	Field of application
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DC72921	COE2-2hexyl	COE2-2hexyl represents an innovative class of antimicrobial agents, demonstrating broad-spectrum antibacterial activity through its unique conjugated oligoelectrolyte (COE) structure.
DC72568	Cymal-6	Cymal-6 (Cyclohexyl-hexyl-β-D-maltoside) is a potent TEM-1 beta-lactamase inhibitor with an Ki value of 40.05 µM. Cymal-6 (Cyclohexyl-hexyl-β-D-maltoside) can be used as glycosidic surfactant.
DC72280	PNU-101603	PNU-101603 is a metabolite of Sutezolid. PNU-101603 has excellent activity against Mycobacterium tuberculosis (MTB).
DC72279	MRV03-070	MRV03-070 is an inhibitor of colibactin-activating peptidase ClbP with an IC50 value of 69 nM, acts like biosynthetic precursor precolibactin.
DC72144	TH-Z145	TH-Z145, a lipophilic bisphosphonate, is a FPPS inhibitor (IC50: 210 nM).
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DC71474	VP-4604	VP-4604 is a potent anti-methicillin-resistant Staphylococcus aureus (MRSA) agent. VP-4604 exhibits significant microbial growth inhibition toward Staphylococcus aureus (ATCC 43300) with MIC of 4-8 µg/mL. VP-4604 inhibits the growth of methicillin‐resistant Staphylococcus aureus with growth inhibition >95%.
DC71466	EDA-DA	EDA-DA is an unnatural dipeptide building block (an ethynyl-D-alanine and a D-alanine). It incorporates a biorthogonal alkyne group into peptidoglycan (PG) through MurF in the cytoplasmic pathway, which enables selective labeling via a click-chemistry reaction. EDA-DA allows labeling of PG in Gram-positive (B. subtilis), Gram-negative (E. coli and C. trachomatis), Mycobacterium (M. smegmatis) and moss plastids (P. patens) with azide modified fluorescent dyes such as Alexa Fluor 488.