Rebamipide mofetil|CAS 1527495-76-6|DC Chemicals

Cas No.:	1527495-76-6
Chemical Name:	Rebamipide mofetil
Synonyms:	Rebamipide mofetil;Rebamipide mofetil [INN];2-morpholin-4-ylethyl 2-[(4-chlorobenzoyl)amino]-3-(2-oxo-1H-quinolin-4-yl)propanoate;2-Morpholin-4-ylethyl 2-(4-chlorobenzoylamino)-3-(2-oxo-1,2-dihydroquinolin-4-yl)propionate;4-Quinolinepropanoic acid, alpha-((4-chlorobenzoyl)amino)-1,2-dihydro-2-oxo-, 2-(4-morpholinyl)ethyl ester
SMILES:	ClC1C([H])=C([H])C(=C([H])C=1[H])C(N([H])C([H])(C(=O)OC([H])([H])C([H])([H])N1C([H])([H])C([H])([H])OC([H])([H])C1([H])[H])C([H])([H])C1=C([H])C(N([H])C2=C([H])C([H])=C([H])C([H])=C12)=O)=O
Formula:	C₂₅H₂₆ClN₃O₅
M.Wt:	483.9440
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:	Rebamipide mofetil is an orally active prodrug of Rebamipide (OPC12759). Rebamipide is a mucoprotective agent. Rebamipide induces COX-2 expression, increases PGE2 levels, and enhances gastric mucosal defense in a COX-2-dependent manner[1].
References:	[1]. Cho, Eui Hwan, et al.Pharmaceutical composition comprising rebamipide precursor for oral administration for preventing or treating immune disease and metabolic disease.WO2017138717A1.

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