AC264613 is a potent and selective protease-activated receptor 2 (PAR2) agonist (pEC50 = 7.5). Displays no activity at other PAR subtypes and exhibits no significant activity at over 30 other receptors implicated in nociception and inflammation.

A Tyrosine kinase inhibitor.

A potent, specific, orally active melanin concentrating hormone receptor 1 (MCHR1) inhibitor with kI of 3.8 nM, >100-fold selectivity over a battery of GPCRs, ion channels and enzymes.

A novel potent, selective Sirt2 inhibitor with IC50 of 3.745 uM.

A cell permeable, mechanistically unique inhibitor of protein sumoylation.

5S rRNA modificator is a suitable electrophile for 2’-hydroxyl acylation on structured RNA molecules, yielding accurate structural information comparable to that obtained with existing probes; 5S rRNA RNA modification.

3,4-Dicaffeoylquinic acid (3,4-DCQA) is a polyphenol with diverse biological activities.