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| Cat. No. | Product Name | Field of Application | Chemical Structure |
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| DC23981 | BCX-1470 methanesulfonate Featured |
A serine protease inhibitor that inhibits the esterolytic activity of factor D (IC50=96 nM) and C1s (IC50=1.6 nM).
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| DC10474 | GBT-440(Voxelotor) Featured |
GBT-440(Voxelotor) is a novel small molecule hemoglobin modifier which increases hemoglobin oxygen affinity.
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| DC20309 | ANTISAUVAGINE-30 Featured |
A potent, selective and competitive corticotropin-releasing factor CRF2 receptor antagonist with Ki of 1.4 nM, 100-fold selectiivity over CRF1.
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| DCAPI1056 | Nattokinase Featured |
Nattokinase, Natto fermentation is a potent fibrinolytic enzyme. Nattokinase can break down blood clots by directly hydrolyzing fibrin and plasmin substrate. Nattokinase can be used for the research of cardiovascular diseases.
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| DC32887 | NNC63-0532 Featured |
NNC63-0532 is a potent and selective non-peptide agonist of the NOP receptors.
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| DC26004 | delta-Valerobetaine (hydrobromide) Featured |
Delta-Valerobetaine (hydrobromide) is a precursor of trimethylamine N-oxide (TMAO).
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| DC23380 | TRIM24 inhibitor X Featured |
TRIM24 inhibitor X is a potent TRIM24 bromodomain inhibitor for synthesis dTRIM24..
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| DC22843 | DDX3-IN-16d Featured |
A small molecule inhibitor (IC50=0.3 uM) of DEAD-box polypeptide 3 (DDX3), a human host factor required for the replication of several DNA and RNA viruses.
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| DCC4088 | Pf-06424439 Mesylate Featured |
Potent and selective inhibitor of diacylglycerol acyltransferase 2 (DGAT2)
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| DC74133 | PSB-CB-27 Featured |
PSB-CB-27 is a potent, selective antagonist of GPR18 with IC50 of 650 nM, shows no inhibition on GPR55 and low affinity for CB1/CB2 receptors.
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| DC46883 | Tinlarebant Featured |
Tinlarebant (LBS-008) is an orally active non-retinoid RBP4 (retinol-binding protein 4) antagonist. Tinlarebant can be used for the research of the Stargardt disease.
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| DCC0543 | Alk-001 Featured |
ALK-001 is a vitamin A analog potentially for the treatment of Stargardt’s disease.
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| DC74185 | SS-1-148 Featured |
SS-1-148 is a potent, selective inhibitor of human ornithine δ-aminotransferase (hOAT) with Ki of 60 uM, shows excellent selectivity over other related aminotransferases (e.g., GABA-AT).
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| DC12091 | AdipoRon hydrochloride Featured |
AdipoRon hydrochloride is an orally active and specific AdipoR agonist, binding to AdipoR1 and AdipoR2, with Kds of 1.8 and 3.1 μM, respectively.
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| DC7049 | AdipoRon Featured |
AdipoRon is a novel small-molecule AdipoR agonist; binds to both AdipoR1(Kd= 1.8 uM) and AdipoR2(Kd=3.1 uM).
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| DC47318 | 7,12-Dimethylbenz[a]anthracene (DMBA) Featured |
7,12-Dimethylbenz[a]anthracene (DMBA) is an immunosuppressor as well as a potent organ-specific carcinogen.
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| DCAPI1014 | Eplerenone Featured |
Eplerenone, also known as Inspra and CGP-30083, is a selective aldosterone receptor antagonist used to treat hypertension and congestive heart failure. Eplerenone provides marked protection against vascular injury in the kidney and heart.
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| DC74064 | Macrocyclic peptide D4-2 Featured |
Macrocyclic peptide D4-2 is a macrocyclic peptide consisting of 15 amino acids that binds to the ectodomain of mouse SIRPα (Kd=10 nM, IgV-B6 SIRPα) and efficiently blocks CD47-SIRPα interaction in an allosteric manner (IC50=0.18 uM).
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| DC26215 | GsMTx-4 Featured |
#N/A
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| DC49967 | (Rac)-RP-6306 Featured |
Myt1-IN-4 (compound 181) is a potent Myt1 inhibitor with an IC50 of <10 nM. Myt1-IN-4 has anticancer effects.
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| DC71835 | (R)-RP-6306 Featured |
(R)-RP-6306 (183) can be used for the research of Myt1 mediated diseases and kinds of cancer for slowing the progression of cancer.
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| DC22654 | MMV-667492 Featured |
MMV-667492 (MMV 667492, MMV667492) is a novel potent Ezrin inhibitor with Kd of 29.4 nM.
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| DC12624 | RAS activator compound 1 Featured |
RAS activator compound 1 is a small molecule RAS activator compound that increases the rate of SOS-catalyzed nucleotide exchange in vitro with EC50 of 14 uM; targets SOS1 induced biphasic modulation of RAS-GTP and ERK phosphorylation levels, through negative feedback on SOS1 that regulates the interaction between SOS1 and GRB2.
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| DC23789 | AK778 Featured |
AK778 (Col001) is a small-molecule compound that inhibits the interaction of Hsp47 with collagen, competitively inhibits the interaction and causes the inhibition of collagen secretion by destabilizing the collagen triple helix. .
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| DC20439 | LXRβ agonist 17 Featured |
LXRβ agonist 17 is a novel, potent, orally active liver X receptor β (LXRβ) agonist with Ki/EC50 of 3/21 nM, displays 27-fold selectivity over LXRα; also exhibits excellent selectivity against other nuclear hormone receptors (>3,000-fold); induces the expression of LXR target genes in vitro and in vivo.
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| DC22537 | SMAP Featured |
SMAP (DT-061, DT061) is an orally bioavailable small molecule activator of PP2A, inhibits KRAS-driven tumor growth.
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| DC46349 | ALS-I Featured |
ALS-I, an acid-Liable surfactant, is adopted for in-solution enzymatic digestions, can help to solubilize hydrophobic proteins. ALS-I is significantly enhanced peptide recovery for mass spectrometry (MS) mapping in the study of the proteomes of regenerating rat retina and mouse brain.
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| DC40519 | BMS-986235 Featured |
BMS-986235 (LAR-1219) is a selective, orally active formyl peptide receptor 2 (FPR2) agonist, with EC50s of 0.41 nM and 3.4 nM for hFPR2 and mFPR2, respectively. BMS-986235 has potential for the prevention of heart failure.
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| DC26078 | GNE-616 Featured |
GNE-616 (GNE616) is a highly potent, metabolically stable, subtype selective inhibitor of Nav1.7 with Ki of 0.79 nM (hNav1.7).
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| DCC1706 | Dd04107 Featured |
Novel inhibitor of α-calcitonin gene-related peptide (α-CGRP) exocytotic release from primary sensory neurons, selectively interacting with Synaptotagmin 1
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