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(±)-U-50488

  Cat. No.:  DC79876   Featured
Chemical Structure
83913-05-7
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More than 5000 active chemicals with high quality for research!
Field of application
(±)-U-50488 ((±)-trans-(1R,2R)-U-50488) is a selective kappa opioid receptor agonist. (±)-U-50488 can improve symptoms related to status epilepticus, but has no significant effect on spontaneous seizure episodes. (±)-U-50488 can be used for research of epilepsy.
Cas No.: 83913-05-7
Chemical Name: TRANS-(+/-)-3,4-DICHLORO-N-METHYL-N-(2-[1-PYRROLIDINYL]CYCLOHEXYL)-BENZENEACETAMIDE METHANESULFONATE SALT
Synonyms: TRANS-(+/-)-3,4-DICHLORO-N-METHYL-N-(2-[1-PYRROLIDINYL]CYCLOHEXYL)-BENZENEACETAMIDE METHANESULFONATE SALT;TRANS-(+/-)-3,4-DICHLORO-N-METHYL-N-(2-[1-PYRROLIDINYL]CYCLOHEXYL)-BENZENEACETAMIDE METHANESUL...;U 50488H;CHEMBL482811;SCHEMBL548872;NCG-C00093883-01;Opera_ID_588;Benzeneacetamide, 3,4-dichloro-N-methyl-N-[(1R,2R)-2-(1-pyrrolidinyl)cyclohexyl]-, methanesulfonate (1:1);MLS000069740;trans-(+/-)-3,4-Dichloro-N-methyl-N-(2-[1-pyrrolidinyl]cyclohexyl)benzeneacetamide methanesulfonate;Lopac-D-8040;U-50488 methane sulfonate;HMS2232L15;2-(3,4-dichlorophenyl)-N-methyl-N-((1R,2R)-2-(pyrrolidin-1-yl)cyclohexyl)acetamide methanesulfonate;MLS001076340;83913-05-7;2-(3,4-dichlorophenyl)-N-methyl-N-[(1R,2R)-2-pyrrolidin-1-ylcyclohexyl]acetamide;methanesulfonic acid;DTXSID301004058;(+/-)-trans-U-50488 methanesulfonate salt;83913-06-8;SMR000058892;Benzeneacetamide, 3,4-dichloro-N-methyl-N-(2-(1-pyrrolidinyl)cyclohexyl)-, trans-(+-)-, monomethanesulfonate;U50,488H;NCGC00016144-01;trans-(+/-)-3,4-Dichloro-N-methyl-N-[2-(1-pyrrolidinyl)cyclohexyl]benzeneacetamide hydrochloride
SMILES: ClC1=C(C=CC(=C1)CC(N(C)[C@@H]1CCCC[C@H]1N1CCCC1)=O)Cl.S(C)(=O)(=O)O
Formula: C20H30Cl2N2O4S
M.Wt: 465.43
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
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DC79876 (±)-U-50488 (±)-U-50488 ((±)-trans-(1R,2R)-U-50488) is a selective kappa opioid receptor agonist. (±)-U-50488 can improve symptoms related to status epilepticus, but has no significant effect on spontaneous seizure episodes. (±)-U-50488 can be used for research of epilepsy.
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