AG-1557| cas 189290-58-2|DC Chemicals

Cas No.:	189290-58-2
Chemical Name:	AG-1557
Synonyms:	AG-1557;N-(3-iodophenyl)-6,7-dimethoxyquinazolin-4-amine;AG1557
SMILES:	COC1=C(C=C2C(=C1)C(=NC=N2)NC3=CC=CC(=C3)I)OC
Formula:	C₁₆H₁₄In₃O₂
M.Wt:	407.205735683441
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:	AG-1557, compound 22 (T), is a ATP competitive inhibitor of epidermal growth factor receptor (EGFR) tyrosine kinase with a pIC50 value of 8.194[1].
References:	[1]. Akshada Joshi， et al. Identification of Potential Novel EGFR Inhibitors using a Combination of Pharmacophore and Docking Methods. International Journal of Pharmacy and Pharmaceutical Sciences, ISSN- 0975-1491 Vol 7, Issue 6, 2015

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