AZD6280|CAS 942436-93-3|GABAA receptor modulator

Cas No.:	942436-93-3
Chemical Name:	4-amino-8-(2,5-dimethoxyphenyl)-N-propyl-3-cinnolinecarboxamide
Synonyms:	AZD 6280,AZD-6280
SMILES:	CCCNC(=O)c1c(c2cccc(c2nn1)c3cc(ccc3OC)OC)N
Formula:	C₂₀H₂₂N₄O₃
M.Wt:	366.421
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:	AZD-6280 is a selective GABAA(α2/3) receptor modulator, used for treatment of generalized anxiety disorder.
References:	[1]. Te Beek ET, et al. The effects of the nonselective benzodiazepine lorazepam and the α2 /α3 subunit-selective GABAA receptor modulators AZD7325 and AZD6280 on plasma prolactin levels. Clin Pharmacol Drug Dev. 2015 Mar;4(2):149-54. doi: 10.1002/cpdd.134. Epub 2014 Aug 28.

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