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Cereblon Ligand-Linker Conjugates 9(E3 Ligase Ligand-Linker Conjugates 2)

  Cat. No.:  DC26126   Featured
Chemical Structure
1818885-63-0
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More than 5000 active chemicals with high quality for research!
Field of application
Pomalidomide-PEG4-Ph-NH2 is a synthesized E3 ligase ligand-linker conjugate that incorporates the Pomalidomide based cereblon ligand and 4-unit PEG linker used in PROTAC technology.
Chemicals PropertiesBiological activity Related products COA MSDS Datasheet
Cas No.: 1818885-63-0
SMILES: O=C1N(C(CC2)C(NC2=O)=O)C(C3=C1C=CC=C3NCCOCCOCCOCCOC4=CC=C(N)C=C4)=O
Formula: C27H32N4O3
M.Wt: 540.57
Purity: >98%
Description: E3 Ligase Ligand-Linker Conjugates 2 incorporates a ligand for the E3 ubiquitin ligase, and a PROTAC linker, which bring together target protein and ubiquitinating machinery.
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