ML267 TFA |cas 1542213-67-1|DC Chemicals

Cas No.:	1542213-67-1
Chemical Name:	4-(3-chloro-5-(trifluoromethyl)pyridin-2-yl)-N-(4-methoxypyridin-2-yl)piperazine-1-carbothioamide trifluoroacetate
Synonyms:	MLS003874059;SMR002530704;4-(3-Chloro-5-(trifluoromethyl)pyridin-2-yl)-N-(4-methoxypyridin-2-yl)piperazine-1-carbothioamide 2,2,2-trifluoroacetate;4-(3-chloro-5-(trifluoromethyl)pyridin-2-yl)-N-(4-methoxypyridin-2-yl)piperazine-1-carbothioamide trifluoroacetate;ML267
SMILES:	ClC1=CC(C(F)(F)F)=CN=C1N1CCN(C(NC2C=C(C=CN=2)OC)=S)CC1.FC(C(=O)O)(F)F
Formula:	C₁₉H₁₈ClF₆N₅O₃S
M.Wt:	545.89
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

ML267 a potent Sfp phosphopantetheinyl transferase (PPTases) inhibitor with an IC50 of 0.29 μM. ML267 also inhibits AcpS-PPTase with an IC50 of 8.1 μM. ML267 possesses specific Gram-positive-targeted bactericidal activities.

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