BUN79398|cas 2377379-39-8|DC Chemicals

Cas No.:	2377379-39-8
Chemical Name:	N-(2-(1-aminoisoquinolin-6-yloxy)-4-methylphenyl)-2-methoxybenzenesulfonamide
Synonyms:	MRGPRX1 agonist 1; BUN79398; BUN-79398; BUN 79398;
SMILES:	O=S(C1=CC=CC=C1OC)(NC2=CC=C(C)C=C2OC3=CC4=C(C(N)=NC=C4)C=C3)=O
Formula:	C₂₃H₂₁N₃O₄S
M.Wt:	435.498
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

BUN79398(MRGPRX1 agonist 1) is a highly potent agonist of MRGPRX1 (Mas-related G-protein-coupled receptor X1), with an EC50 of 50 nM, and is inactive on MRGPRC11. Analgesic effect[1].

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