GD20|cas |DC Chemiclas

Cas No.:
Chemical Name:	GD20
Synonyms:	GD 20;GD-20
SMILES:	CCC[C@@H]1NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC2=CC=CC=C2)NC(=O)[C@H](C)NC(=O)[C@H](CC2=CNC3=CC=CC=C23)NC(=O)[C@H](CCC(N)=O)NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CC2=CC=CC=C2)NC(=O)[C@H]([C@@H](C)O)NC(=O)[C@H]([C@@H](C)CC)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](CC2=CC=C(O)C=C2)NC(=O)CSCC(C(=O)NCC(N)=O)NC(=O)[C@@H]2CCCN2C1=O
Formula:	C₈₉H₁₂₄O₂₀N₂₂S
M.Wt:	1854.16
Purity:	>98%

Description:

GD20 is a cell-permeable, nucleotide-inactive-state-selective inhibitor of Gαs, with high selectivity over other G protein subfamilies. GD20 inhibits Gαs steady-state GTPase activity with IC50 of 1.15 μM.

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