(R)-69|cas |DC Chemicals

Cas No.:
Chemical Name:	(R)-69
SMILES:	C[C@@H]1C=C(C2=CNC3=C2C=CC=N3)CNC1
Formula:	C₁₃H₁₅N₃
M.Wt:	213.28
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

(R)-69 is a 5-HT2AR partial agonists with EC50 of 41 nM, and shows 4.6-fold/29-fold selectivity over 5HT2BR/5HT2CR. (R)-69 has substantial brain permeability in mouse pharmacokinetic studies and dose not possess locomotor-stimulating or reinforcing activity.

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