GSK-2894631A|GSK2894631A

Cas No.:	2101626-26-8
SMILES:	C1C2=CC=C(OC(F)F)C=C2N=CC=1C(N[C@@H]1CC[C@@H](C(O)(C)C)CC1)=O
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:	GSK-2894631A(HPGDS inhibitor 2) is a highly potent and selective hematopoietic prostaglandin D synthase (H-PGDS) inhibitor with an IC50 of 9.9 nM[1].
Target:	IC50: 9.9 nM (H-PGDS)[1]
References:	[1]. Deaton DN, et al. The discovery of quinoline-3-carboxamides as hematopoietic prostaglandin D synthase (H-PGDS) inhibitors. Bioorg Med Chem. 2019 Apr 15;27(8):1456-1478.

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GSK-2894631A(HPGDS inhibitor 2)