Cruzain-IN-1|ML092

Cas No.:	1199523-24-4
SMILES:	CCN1C2=NC(C#N)=NC(NC3=CC(F)=CC(F)=C3)=C2N=C1
Formula:	C₁₄H₁₀F₂N₆
M.Wt:	300.27
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:	Cruzain-IN-1 is a covalent and reversible Cruzain inhibitor, with an IC50 of 10 nM.
Target:	IC50:10 nM (Cruzain)[1].
References:	[1]. Lee GM, et al. Mapping inhibitor binding modes on an active cysteine protease via nuclear magnetic resonance spectroscopy. Biochemistry. 2012 Dec 18;51(50):10087-98.

Cat. No.	Product name	Field of application
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DC37321	AI3-15902	AI3-15902 is a biochemical.
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DC37245	Piperonyl butoxide	Piperonyl butoxide (PBO) is an organic compound used as a component of pesticide formulations. It is a waxy white solid. It is a synergist. That is, despite having no pesticidal activity of its own, it enhances the potency of certain pesticides such as carbamates, pyrethrins, pyrethroids, and rotenone.[1] It is a semisynthetic derivative of safrole.
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Cruzain-IN-1（ML092）