PF-06256142|PF06256142

Cas No.:	1609583-14-3
Chemical Name:	(+)-4-(3-Methyl-4-(6-methylimidazo[1,2-a]pyrazin-5-yl)phenoxy)furo[3,2-c]pyridine
Synonyms:	PF06256142
SMILES:	C(OC1=CC=C(C2N3C=CN=C3C=NC=2C)C(C)=C1)1=NC=CC2OC=CC1=2
Formula:	C₂₁H₁₆N₄O₂
M.Wt:	356.385
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

PF-06256142 (PF06256142) is a potent and selective orthosteric agonist of the D1 receptor with EC50 (cAMP) of 33 nM, shows exquisitely selectivity over D2; demonsrates reduced receptor desensitization relative to dopamine and other catechol-containing agonists.

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