STK321130（FLT3-IN-2）|FLT3 inhibitor|CAS 923562-23-6

Cas No.:	923562-23-6
Chemical Name:	5-[(5-Chloro-1H-pyrrolo[2,3-b]pyridin-3-yl)methyl]-N-[[4-(trifluoromethyl)phenyl]methyl]-2-pyridinamine
Synonyms:	AKR1C3 Inhibitor 5f
SMILES:	FC(C1=CC=C(CNC2=NC=C(CC3=CNC4=NC=C(Cl)C=C43)C=C2)C=C1)(F)F
Formula:	C₂₁H₁₆ClF₃N₄
M.Wt:	416.1
Purity:	>98%
Sotrage:	4°C for 1 year, -20°C for more than 2 years

Description:	STK321130（FLT3-IN-2) is a FLT3 inhibitor with IC50 of ＜ 1 μM, detailed information refer to WO 2012158957 A2 and WO 2007013896.
References:	[1]. Zhang, Chao, et al. Kinase modulation for the treatment of leukemias. From PCT Int. Appl. (2012), WO 2012158957 A2 20121122. [2]. Zhang Chao, et al. 7-Azaindole derivatives and their preparation, pharmaceutical compositions and use for modulating c-kit and c-fms activity. From PCT Int. Appl. (2007), WO 2007013896 A2 20070201.

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STK321130（FLT3-IN-2)