TCS 5861528|TRPA1 channel blocker|DC Chemials

Cas No.:	332117-28-9
Chemical Name:	2-(1,3-Dimethyl-2,6-dioxo-1,2,3,6-tetrahydro-7H-purin-7-yl)-N-[4-(1-methylpropyl)phenyl]acetamide
Synonyms:	TCS 5861528,TCS-5861528,TCS5861528
SMILES:	CCC(C)C1=CC=C(C=C1)NC(=O)CN2C=NC3=C2C(=O)N(C(=O)N3C)C
Formula:	C₁₉H₂₃N₅O₃
M.Wt:	369.42
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

TCS 5861528 is a TRPA1 channel blocker that antagonizes AITC- and 4-HNE-evoked calcium influx (IC50 values are 14.3 and 18.7μM respectively).

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