ATR inhibitor 4|CAS 2417489-10-0|DC Chemicals

Cas No.:	2417489-10-0
Chemical Name:	8-Oxabicyclo[3.2.1]octan-3-ol, 3-[6-[(3R)-3-methyl-4-morpholinyl]-1-(1H-pyrazol-3-yl)-1H-pyrazolo[3,4-b]pyridin-4-yl]-, (3-endo)-
Synonyms:	8-Oxabicyclo[3.2.1]octan-3-ol, 3-[6-[(3R)-3-methyl-4-morpholinyl]-1-(1H-pyrazol-3-yl)-1H-pyrazolo[3,4-b]pyridin-4-yl]-, (3-endo)-;RP-3500;RP-3500 (Synonyms: ATR inhibitor 4);Camonsertib
SMILES:	OC1(CC2CCC(O2)C1)C1C=C(N2CCOCC2C)N=C2N(C3=NNC=C3)N=CC=12
Formula:	C₂₁H₂₆N₆O₃
M.Wt:	410.47
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:	ATR inhibitor 4 (compound 121) is a potent ATR inhibitor. ATR inhibitor 4 has antitumor activity.
Target:	ATR
References:	[1]. Maria Koehler, et al. Use of atr inhibitors in combination with parp inhibitors. WO2021119523A1

Cat. No.	Product name	Field of application
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DC47131	ATR inhibitor 4	ATR inhibitor 4 (compound 121) is a potent ATR inhibitor. ATR inhibitor 4 has antitumor activity.
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DC9309	AZD-0156	AZD-0156 is an orally bioavailable ataxia telangiectasia mutated (ATM) kinase inhibitor, with potential chemo-/radio-sensitizing and antineoplastic activities.