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GTX-134

Cat. No.: DC74417

Chemical Structure

1356059-82-9

For research use only. We do not sell to patients.

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Field of application

GTx-134 (GTx 134) is a selective small-molecule inhibitor of IGF-1R and insulin receptor (IR) with biochemical IC50 of 97 nM and 187 nM, respectively.

Chemicals Properties Biological activity Related products COA MSDS Datasheet

Cas No.:	1356059-82-9
Chemical Name:	GTX-134
Formula:	C₃₃H₄₀N₆O₆S
M.Wt:	648.78

Cat. No.	Product name	Field of application
DC74417	GTX-134	GTx-134 (GTx 134) is a selective small-molecule inhibitor of IGF-1R and insulin receptor (IR) with biochemical IC50 of 97 nM and 187 nM, respectively.
DC74416	BM001	BM001 (BM-001) is a small molecular inhibitor of the integral growth hormone/insulin-like growth factor-1 (GH/IGF1) axis, shows potent antiproliferative effect on cancer cells MDA-MM-231 and Colo-205 with IC50 of 20-30 nM.
DC50117	AZ12253801	AZ12253801 is an ATP-competitive IGF-1R tyrosine kinase inhibitor that shows ∼10-fold selectivity over the insulin receptor. AZ12253801 inhibits IGF-1R–driven proliferation in 3T3 mouse fibroblasts (transfected with human IGF-1R) with an IC50 of 17 nmol/L. The IC50 for epidermal growth factor receptor (EGFR)–driven proliferation is 440 nmol/L. Anti-tumor activity.

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