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ibap

  Cat. No.:  DC55001   Featured
Chemical Structure
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More than 5000 active chemicals with high quality for research!
Field of application
iBAP (BAP1 inhibitor I) is a first-in-class inhibitor of the catalytic activity of BAP1 histone H2A deubiquitinase complex with IC50 of 0.5-1 uM in vitro,
Chemicals PropertiesBiological activity Related products COA MSDS Datasheet
Cas No.:
Chemical Name: ibap
Synonyms: I-BAP
Formula: C18H16N2O2
M.Wt: 292.12
Purity: >97%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Publication: Lu Wang et al, Epigenetic targeted therapy of stabilized BAP1 in ASXL1 gain-of-function mutated leukemia, Nature Cancer (2021). DOI: 10.1038/s43018-021-00199-4
Description: iBAP (BAP1 inhibitor I) is a first-in-class inhibitor of the catalytic activity of BAP1 histone H2A deubiquitinase complex with IC50 of 0.5-1 uM in vitro,
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