Fascaplysin (chloride)|cas 119391-56-9|DC Chemicals

Cas No.:	119391-56-9
Chemical Name:	mAChR-IN-1
Synonyms:	mAChR-IN-1
SMILES:	O=C(C(C1CCN(CC2=CC=C(I)C=C2)CC1)(C3=CC=CC=C3)CC4)NC4=O
Formula:	C₂₃N₂O₂IH₂₅
M.Wt:	488.3613
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:	mAChR-IN-1 is a potent muscarinic cholinergic receptor(mAChR) antagonist with IC50 of 17 nM.
References:	[1]. Wilson AA, et al. Synthesis and biological evaluation of [125I]- and [123I]-4-iododexetimide, a potent muscarinic cholinergic receptor antagonist. J Med Chem. 1989 May;32(5):1057-62.

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mAChR-IN-1