CCG-63802|cas 620112-78-9|DC Chemicals

Cas No.:	620112-78-9
Synonyms:	CCG 63802; CCG63802
SMILES:	N#C/C(C1=NC2=CC=CC=C2S1)=CC3=C(N=C4C(C)=CC=CN4C3=O)OC5=CC=CC(C)=C5
Formula:	C₂₆H₁₈N₄O₂S
M.Wt:	450.5117
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

CCG-63802 is a reversible inhibitor of regulator of G-protein signaling (RGS) protein; with greatest potency at RGS4. CCG-63802 is selective amongst RGS proteins, with greatest potency at RGS4. CCG-63802 inhibits GTPase accelerating protein activity of RGS4 and blocks its interaction with Gαo. Retains activity under reducing conditions.

Cat. No.	Product name	Field of application
DC9613	CCG-63808	CCG-63808 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins.
DC9612	CCG-63802	CCG-63802 is a reversible inhibitor of regulator of G-protein signaling (RGS) protein; with greatest potency at RGS4. IC50 value: Target: RGS CCG-63802 is selective amongst RGS proteins, with greatest potency at RGS4.
DC11662	CCG-4986	A non-peptide, selective RGS4 inhibitor that inhibits RGS4/Gα(o) binding with 3 to 5 uM potency.