Novel potent sPLA2 inhibitor, selectively targeting hGIIA and hGIID

Sterol Biosynthesis Inhibitor, Fungicide

Novel p53 Stabilizer for Brain Cell Differentiation

Novel selective orally bioavailable inhibitor of p300/CBP histone acetyltransferase

Novel gamma-secretase modulator

Antibiotic, binding to the bacterial 30S ribosomal subunit, interfering with the initiation of protein synthesis and with proper protein elongation and leading to bacterial cell death

Novel anti-tuberculosis agent against intracellular Mycobacterium tuberculosis

Novel photo-controllable hydrogen sulfide donor applicable in live cells

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Novel telomerase inhibitor

Novel Programmed Death Ligand 1 (PD-L1) Binding Peptide (a Peptide Ligand for PD-L1)

Sorting inhibitor, blocking Vps16 function, one protein in the class C tethering complex, and increasing aflatoxin synthesis and export

Novel partial inhibitor of amphetamine-induced dopamine release

DAT modulator, being unique in affecting substrate uptake without impacting efflux

Human norepinephrine transporter blocker

Natural inhibitor of the Kv1.3 channels in a concentration-dependent manner

Inhibitor of constitutive and inducible STAT3 activation through the activation of SHP-2 tyrosine phosphatase

Natural analgesic, antipyretic, anti-inflammatory, and anti-tumor agent

A2A adenosine receptor agonist

Novel, selective and orally bioavailable c-Met inhibitor, exhibiting antitumor activity both in vitro and in vivo

Novel potent and selective allosteric modulator of sigma-1 receptor

Unique somatostatin receptor subtypes 2-, 4- and 5-selective analogue, effectively reducing GH secretion in human GH-secreting pituitary adenomas even in Octreotide non-responsive tumours.

Novel long-acting, reversible albumin-binding growth hormone (GH) derivative for treatment of growth hormone dificiency

Novel oral, broad-spectrum matrix metalloproteinase inhibitor (MMPI), being >10-fold more active than marimastat in inhibiting the processing of cell-bound TNF-alpha

Natural tumor antagonistic steroidal alkaloid, inducing typical cellular apoptotic hallmarks and cell cycle blockage at S-G2/M phase, activating nuclear import of DFF-40 mediated nucleosomal disruption and cell demise

Narcolepsy agent, being used to treat catalepse and daytime sleepiness in patients with narcolepsy

Hepatoprotective and choleretic agent

PPARdelta receptor agonist

Novel potent inhibitor of SOD1-Derlin-1 interaction

Novel potent inhibitor of SOD1-Derlin-1 interaction