Moderate alpha-l-fucosidase inhibitor

Natural microbial metabolite of isoflavone genistein, increasing the lifespan and improving the thermal and oxidative stress tolerance of C. elegans

Less active enantiomer of Elexacaftor

BAY-805 is a potent and selective USP21 inhibitor. BAY-805 is a non-covalent inhibitor with low nanomolar affinity for USP21 and high selectivity over other DUB targets as well as kinases, proteases, and other common off-targets.

Metabolite of VX-740

Vesicular monoamine transporter-2 (VMAT2) inhibitor, with 15-​fold greater affinity than GZ-​793A

Inactive control for VinSpinIn

Negative control for EED inhibitor EED226

Negative control compound for UNC3866 which is a potent antagonist of the methyllysine (Kme) reading function of the Polycomb CBX and CDY families of chromodomains

FIT-039 is a potent, selective CDK9 inhibitor with IC50 of 5.8 uM for CKD9/cyclin T1, suppresses the replication of HSV-1 (IC50=0.69 uM).

Negative control for UCSF924

Cell impermeant homolog of UCD38B, inhibitor of uPA (urokinase plasminogen activator)

Negative control for TP-004

Negative control for TP-238

Negative control for TP-040

Negative control for THPP-1

Novel potent and selective NUDT15 inhibitor (MG IC50 = 35 nM), potentiating the anti-HCMV efficacy of ganciclovir

Negative control for TH1760

Metabolite of Telmisartan

Novel novel anti-tuberculosis (TB) agent, possessing improved safety properties compared to bedaquiline

Cell permeable Cx43 hemichannel blocker, being used a control peptide for TAT-Gap19

Negative control for T3-CLK

Prodrug of ADAM17 inhibitor SN-4

Negative control for SGC-STK17B-1, showing IC50 > 10,000 nM against STK17B

Negative control for SGC-CLK-1

Negative control for SGC-CK2-1

Negative control for SGC-CAMKK2-1

Negative control for SGC-SMARCA-BRDVIII

Novel cell permeable CD45 phosphatase inhibitor; Prodrug of RWJ-60475

Metabolite of ozanimod, exhibiting a similar specificity profile as ozanimod at the S1P receptor family in vitro and pharmacodynamic profile in vivo