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| Cat. No. | Product Name | Field of Application | Chemical Structure |
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| DC8602 | LY311727 Featured |
LY 311727 is a specific group II sPLA2 (phospholipase A2 (PLA2)) inhibitor which has been reported to attenuate VEGF-mediated platelet-activating factor (PAF) synthesis in HUVEC and BAEC cells.
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| DC8697 | Terbuthylazine Featured |
Terbuthylazine is an inhibitor of acetolactate syntase (ALS), is a selective herbicide.
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| DC8684 | Fenoxaprop-P-ethyl Featured |
Fenoxaprop-P-ethyl is a post-emergent phenoxy herbicide of the aryloxyphenoxy propionate group.
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| DC10569 | MDK1088(T.cruzi Inhibitor) Featured |
MDK-1088, also known as T.cruzi Inhibitor, is a Trypanosoma cruzi inhibitor. MDK-1088 has CAS#1350920-22-7 . The last 4 digit f CAS# was used in its name.
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| DC10573 | MDK34597 (PI3K inhibitor) Featured |
MDK34597 is a PI3K inhibitor.MDK34597 is an analog of PI-103 and acts as a dual PI3K/mTOR Inhibitor.
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| DC10572 | MDK35833(Oct3/4-inducer-1) Featured |
MDK35833, also known as Oct3/4-inducer-1, is a potent Oct3/4-inducer.
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| DC24209 | MDK7229(MD2-IN-1) Featured |
MDK7229, also known as MD2-IN-1 is a MD2 (Myeloid differentiation protein 2) inhibitor.
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| DC10570 | MDK74978(Multi-kinase inhibitor) Featured |
MDK74978, also known as Multi-kinase inhibitor I, is a Multi-kinase inhibitor. MDK74978 has CAS#778274-97-8. The last 5 digit was used in its name.
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| DC10571 | MDK-8582(Hnps-PLA Inhibitor) Featured |
MDK-8582, also known as Hnps-PLA Inhibitor, is an nhibitor of human nonpancreatic secretory Phospholipase A (hnps-PLA).
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| DC10650 | MDVN1003 Featured |
MDVN1003 is a potent inhibitor of BTK amd PI3K delta.
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| DC8712 | Deoxycorticosterone acetate Featured |
Deoxycorticosterone acetate is a steroid hormone produced by the adrenal gland that possesses mineralocorticoid activity and acts as a precursor to aldosterone.
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| DC8906 | Indinavir Featured |
Indinavir(MK-639; L735524) is a potent and specific HIV protease inhibitor that appears to have good oral bioavailability.
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| DC8910 | Flunarizine dihydrochloride Featured |
Flunarizine is a selective calcium entry blocker.
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| DC8932 | TG003 Featured |
TG003 is a potent and ATP-competitive Cdc2-like kinase (Clk) inhibitor with IC50 of 20 nM, 200 nM, and 15 nM for Clk1, Clk2, and Clk4, respectively. No inhibitory effect on Clk3, SRPK1, SRPK2, or PKC.
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| DC8939 | Tolrestat Featured |
Tolrestat(AY-27773) is a potent, orally active aldose reductase inhibitor with IC50 value of 35 nM.
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| DC9375 | GPDA Featured |
GPDA(Glycylproline p-nitroanilide tosylate) is the substarate of X-Prolyl dipeptidyl-aminopeptidase in the enzyme assay.
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| DC9460 | CHR-6494 Featured |
CHR-6494 is a potent and selective Haspin (Haploid Germ Cell-Specific Nuclear Protein Kinase) inhibitor that blocks H3T3ph phosphorylation.
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| DC9500 | Cevimeline (hydrochloride hemihydrate) Featured |
Cevimeline hydrochloride hemihydrate, a novel muscarinic receptor agonist, is a candidate therapeutic drug for xerostomia in Sjogren's syndrome.
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| DC9569 | Nefazodone (hydrochloride) Featured |
Nefazodone hydrochloride is an antidepressant drug.
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| DC9651 | Ingenol 3-angelate Featured |
Ingenol 3-Angelate is a PKC(protein kinase C)activator; anti-cancer drug and an active ingredient in Euphorbia peplus.
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| DC8979 | Stavudine Featured |
Stavudine is a nucleoside analog that inhibits reverse transcriptase and has in vitro activity against HIV.
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| DC9010 | Sasapyrine Featured |
Salsalate is a nonsteroidal anti-inflammatory drug (NSAID).
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| DC20065 | PF-06733804 Featured |
Trk-IN-3 is a potent pan-Trk inhibitor in cell-based assays with IC50s of 8.4 nM, 6.2 nM and 2.2 nM for TrkA, TrkB and TrkC, respectively. Anti-hyperalgesic effect.
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| DC20297 | 6-Hydroxy-DL-DOPA Featured |
6-Hydroxy-DL-DOPA is a small-molecule that disrupts with RAD52 oligomerization, inhibits ssDNA binding by RAD52 with IC50 of 1.1 uM and by RAD52 (1 209) with IC50 of 1.6 uM.
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| DC20857 | Calhex-231 Featured |
Calhex-231 is a potent negative allosteric modulator of CaSR that blocks calcium-mediated activation with IC50 of 0.39 uM.
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| DC20945 | DC_AC50 Featured |
DC_AC50 (DCAC50) is a small molecule that inhibits the human copper chaperones Atox1 and CCS (Kd=6.8 and 8.2 uM), blocks copper trafficking and significantly attenuates cancer cell proliferation.
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| DC21002 | Edelfosine Featured |
Edelfosine is a synthetic lysophospholipid analog that selectively inhibits PLC with IC50 of 9.6 uM in fibroblasts and adenocarcinoma cells.
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| DC20866 | CC-671 Featured |
CC-671 is a potent, selective, dual TTK (Mps1)/CLK2 inhibitor with IC50 of 5/3 nM, respectively.
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| DC33031 | CRANAD-2 Featured |
CRANAD-2 is a difluoroboron-derivatized curcumins as near-infrared probe for in vivo detection of amyloid-beta deposits. Upon interacting with Abeta aggregates, CRANAD-2 undergoes a range of changes, which include a 70-fold fluorescence intensity increase, a 90 nm blue shift (from 805 to 715 nm), and a large increase in quantum yield. Moreover, this probe also shows a high affinity for Abeta aggregates (K(d) = 38.0 nM), a reasonable log P value (log P = 3), considerable stability in serum, and a weak interaction with albumin. After intravenous injection of this probe, 19-month-old Tg2576 mice exhibited significantly higher relative signal than that of the control mice over the same period of time.
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| DC33238 | A286982 Featured |
A286982 is an inhibitor that blocks the integrin-ligand interaction between leukocyte function-associated antigen-1 (LFA-1) and intercellular adhesion molecule-1.
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