AZ10606120 dihydrochloride|cas 607378-18-7|DC Chemicals

Cas No.:	607378-18-7
Chemical Name:	AZ10606120 dihydrochloride
Synonyms:	N-[2-[[2-[(2-HYDROXYETHYL)AMINO]ETHYL]AMINO]-5-QUINOLINYL]-2-TRICYCLO[3.3.1.13,7]DEC-1-YLACETAMIDE DIHYDROCHLORIDE;AZ10606120 dihydrochloride
SMILES:	Cl.Cl.OCCNCCNC1C=CC2C(NC(CC34CC5CC(C3)CC(C5)C4)=O)=CC=CC=2N=1
Formula:	C₂₅H₃₆Cl₂N₄O₂
M.Wt:	495.490
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

AZ10606120 is a potent, specific P2X7 receptor antagonist with Kd of 1.4 and 19 nM at human and rat P2X7 receptors respectively; strongly inhibits tumor growth in B16-inoculated C57Bl/6 mice.

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