Cedazuridine|E7727|CAS 1141397-80-9|DC Chemicals

Cas No.:	1141397-80-9
Chemical Name:	Cedazuridine
Synonyms:	E7727;E-7727;E 7727
SMILES:	O=C1N([C@H]2C(F)(F)[C@@H]([C@@H](CO)O2)O)CC[C@@H](O)N1
Formula:	C₉H₁₄F₂N₂O₅
M.Wt:	268.217
Purity:	>95%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:	Cedazuridine (E7727) is a Cytidine Deaminase (CDA) inhibitor with an IC50 value of 0.4 μM[1].
Target:	Cytidine Deaminase (CDA) :IC50: 0.4 μM (CDA)[1]
References:	[1]. Ferraris D, et al. Design, synthesis, and pharmacological evaluation of fluorinated tetrahydrouridine derivatives as inhibitors of cytidine deaminase. J Med Chem. 2014 Mar 27; 57(6):2582-8.

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