MALAT1 inhibitor 5|CAS 827327-28-6|DC Chemicals

Cas No.:	827327-28-6
Chemical Name:	N-(3-methoxybenzyl)-5-(4-methoxyphenyl)-1-methyl-1H-imidazol-2-amine
Synonyms:	MALAT1 inhibitor 5\|Malat1 inhibitor 5
SMILES:	CN1C(C2=CC=C(OC)C=C2)=CN=C1NCC3=CC=CC(OC)=C3
Formula:	C₁₉H₂₁N₃O₂
M.Wt:	323.396
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Publication:	1. Abulwerdi FA, et al. ACS Chem Biol. 2019 Jan 8. doi: 10.1021/acschembio.8b00807.

Description:	MALAT1 inhibitor 5 is a potent and specific Malat1 (Metastasis-associated lung adenocarcinoma transcript 1) inhibitor. MALAT1-IN-1 modulated Malat1 downstream genes in a dose-dependent manner without affecting expression of nuclear enriched abundant transcript 1 (Neat1) [1].
References:	[1]. Abulwerdi FA, et al. Selective Small-Molecule Targeting of a Triple Helix Encoded by the Long Noncoding RNA, MALAT1. ACS Chem Biol. 2019 Feb 15;14(2):223-235.

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MALAT1-IN-1