CMPDA| CAS 380607-77-2

Cas No.:	380607-77-2
Chemical Name:	CMPDA
Synonyms:	CMPDA;[(methylethyl)sulfonyl]{2-[4-(2-{[(methylethyl)sulfonyl]amino}ethyl)phenyl]ethyl}amine
SMILES:	O=S(NCCC1=CC=C(CCNS(=O)(C(C)C)=O)C=C1)(C(C)C)=O
Formula:	C₁₆H₂₈N₂O₄S₂
M.Wt:	376.53452205658
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

CMPDA is a potent positive allosteric modulator of GluR2 receptors with EC50 of 45.4 and 63.4 nM at GluR2i and GluR2o respectively, in a calcium influx screening assays; binds at the modulator binding pocket located at the interdimer interface and the clamshell hinges.

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