MAP4K4-IN-17| CAS 1811510-58-3|DC Chemicals

Cas No.:	1811510-58-3
Chemical Name:	MAP4K4-IN-17
Synonyms:	5-(6-amino-5-(4-chlorophenyl)pyridin-3-yl)pyrimidin-2-amine
SMILES:	NC1=NC=C(C2=CC(C3=CC=C(Cl)C=C3)=C(N)N=C2)C=N1
Formula:	C₁₅H₁₂ClN₅
M.Wt:	297.746
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:	MAP4K4-IN-17 is a potent and highly selective MAP4K4 inhibitor with IC50 of 14.9 nM, showes improved overall drug-like properties compared to PF-06260933; a lead compound for advanced preclinical development.
References:	References 1. Ammirati M, et al. ACS Med Chem Lett. 2015 Oct 6;6(11):1128-33. View Related Products by Target MAP4K

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