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| Cat. No. | Product Name | Field of Application | Chemical Structure |
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| DC2085 | Compound 401 Featured |
Compound 401 is a cell-permeable pyrimido-isoquinolinone compound that acts as a potent, reversible, and ATP-competitive inhibitor of DNA-PK (IC50 = 280 nM) with ~19-fold selectivity over FRAP (mTOR) (IC50 = 5.3 µM).
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| DC10336 | Coenzyme Q9 Featured |
Coenzyme Q9, a nine isoprenyl group-containing member of the ubiquinone family, is a normal constituent of human plasma.
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| DC7106 | Rociletinib (CO-1686) Featured |
CO-1686 is a novel, irreversible and orally delivered kinase inhibitor that specifically targets the mutant forms of EGFR including T790M(IC50=21 nM).
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| DC8095 | Raxatrigine hydrochloride Featured |
CNV1014802(GSK-1014802) is a novel small molecule state-dependent sodium channel blocker; Nav1.7 sodium channel inhibitor.
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| DC23180 | CNV1014802(Raxatrigine) Featured |
CNV1014802 (GSK-1014802, Raxatrigine, Vixotrigine, BIIB074) is a potent, selective Nav1.7 sodium channel blocker, shows analgesic effects and potential in the treatment of cognitive symptoms of schizophrenia in vivo.
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| DC10671 | CNQX disodium salt Featured |
CNQX is a potent AMPA/kainate receptor antagonist. Also antagonist at glycine modulatory site on NMDA receptor complex.
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| DC9799 | CNDAC Featured |
CNDAC is the active component of sapacitabine.
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| DC10752 | CNDAC HCl Featured |
CNDAC (DFP-10917; TAS-109) is an orally available deoxycytosine nucleoside analog with potential antineoplastic activity.
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| DCAPI1428 | Clofarabine Featured |
Clofarabine(Clolar; Clofarex) inhibits the enzymatic activities of ribonucleotide reductase (IC50 = 65 nM) and DNA polymerase. IC50 Value: 65 nM Target: in vitro: Clofarabine is a second generation purine nucleoside analog with antineoplastic activity. It
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| DC7387 | Clemizole Hydrochloride Featured |
Clemizole is a H1 histamine receptor antagonist.Recently, researchers have identified that clemizole hydrochloride can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.
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| DC7668 | CL-387785 Featured |
CL-387785(EKI785; WAY-EKI 785) is an irreversible inhibitor of EGFR with IC50 of 370+/-120 pM; is able to overcome resistance caused by the T790M mutation on a functional level.
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| DC11475 | CK-869 Featured |
CK-869 is an inhibitor of human and bovine actin-related protein 2/3 (Arp2/3) complex.
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| DC12668 | Citarinostat(ACY-241) Featured |
Citarinostat(ACY-241) is a potent, selective and orally available histone deacetylase (HDAC) inhibitor, with potential antineoplastic activity.
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| DC8156 | CIQ Featured |
CIQ is a positive allosteric modulator selective for NR2C/D containing NMDA receptors (EC50 = 2.7 and 2.8 µM for NR2C and NR2D, respectively).
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| DCAPI1372 | Ciprofloxacin (Cipro) Featured |
Ciprofloxacin (Bay-09867) is a fluoroquinolone antibiotic, exhibiting potent antibacterial activity.
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| DC10868 | Cilofexor Featured |
Cilofexor (GS-9674, GS9674) is novel specific, non-steroidal farnesoid X receptor (FXR) agonist that reduces liver fibrosis and ameliorates portal hypertension in rat NASH models.
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| DC7561 | Cilengitide (TFA salt) Featured |
Cilengitide is a potent integrin inhibitor for αvβ3 receptor and αvβ5 receptor with IC50 of 4.1 nM and 79 nM, respectively; ~10-fold selectivity against gpIIbIIIa. Phase 2.
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| DCAPI1021 | Cidofovir(Vistide) Featured |
Cidofovir(Vistide)
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| DC7976 | CID 797718 Featured |
CID-797718 is a compound with unknown details.
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| DC9955 | BCL6 inhibitor(CID5721353) Featured |
CID5721353 is a B-Cell Lymphoma 6 Inhibitor (BCL6 inhibitor).
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| DC7253 | CID-2011756 Featured |
CID-2011756 is a cell-active ATP competitive and specific PKD1 inhibitor that inhibits phorbol ester-induced endogenous PKD1 activation in LNCaP prostate cancer cells.
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| DC10873 | CID16020046 Featured |
CID 16020046 is a potent and selective GPR55(LPI receptor) antagonist; inhibitsGPR55 constitutive activity with IC50 of 0.15 uM.
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| DC2060 | CI994 (Tacedinaline) Featured |
CI994 (Tacedinaline) is an anti-cancer drug which inhibits HDAC1 with IC50 of 0.57 μM.
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| DC8139 | GMX1778(CHS-828) Featured |
CHS-828 is a pyridyl cyanoguanidine anti-tumor agent that has been identified as a competitive inhibitor of Nampt as well as an inhibitor of NF-κB pathway activity.
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| DC8116 | Tosedostat (CHR2797) Featured |
CHR-2797 is an aminopeptidase inhibitor, with IC50 values of 100 nM for LAP3 (LAP), 150 nM for PSAP (PuSA) and 220 nM for CD13 (Aminopeptidase N).
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| DC9082 | Chlorpromazine HCl Featured |
Chlorpromazine Hydrochloride is a dopamine and potassium channel inhibitor used as the prototypical phenothiazine antipsychotic drug.
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| DC7384 | CHIR-98014 Featured |
CHIR-98014 is a potent GSK-3α/β inhibitor with IC50 of 0.65 nM/0.58 nM, with the ability to distinguish GSK-3 from its closest homologs Cdc2 and ERK2.
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| DC9292 | CHIR-090 Featured |
CHIR-090 is a potent LpxC inhibitor, displays two-step time-dependent inhibition and kills a wide range of Gram-negative pathogens as effectively as ciprofloxacin or tobramycin.
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| DC7978 | Tucidinostat(Chidamide) Featured |
Chidamide is a class I HDAC inhibitor with IC50s of 95/160/67/733 nM for HDAC1/2/3/8; also inhibits HDAC10/11(IC50=78/432 nM); no inhibition on HDAC4/5/7/9/6(IC50>30 uM).
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| DC7383 | CH5424802(Alectinib) Featured |
CH5424802(AF 802; Alectinib) is a potent ALK inhibitor with IC50 of 1.9 nM, sensitive to L1196M mutation.
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