HIPK2 inhibitor|cas 1365986-44-2|DC Chemicals

Cas No.:	1365986-44-2
Chemical Name:	Protein kinase inhibitor 1
Synonyms:	Protein kinase inhibitors 1;Protein kinase inhibitors 1 hydrochlorid (1365986-44-2(free base));Protein kinase inhibitor 1
SMILES:	Cl.S1C(NC(/C/1=C/C1=CNC(C(=C1)C1=CN=C(C=C1)N1CCNCC1)=O)=O)=O
Formula:	C₁₈H₁₈ClN₅O₃S
M.Wt:	383.430
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:	Protein kinase inhibitors 1 is a novel inhibitor of HIPK2 with an IC50 of 74 nM and Kd of 9.5 nM.
References:	[1]. Miduturu CV, et al. High-throughput kinase profiling: a more efficient approach toward the discovery of new kinaseinhibitors. Chem Biol. 2011 Jul 29;18(7):868-79.

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Protein kinase inhibitor 1