L-803087 | sst4 Receptor Agonist

Cas No.:	217480-26-7
Chemical Name:	L-Arginine,N2-[4-(5,7-difluoro-2-phenyl-1H-indol-3-yl)-1-oxobutyl]-, methyl ester
Synonyms:	L-Arginine,N2-[4-(5,7-difluoro-2-phenyl-1H-indol-3-yl)-1-oxobutyl]-, methyl ester;L-803,087 TRIFLUOROACETATE;L-803,087 trifluoroacetate,N2-[4-(5,7-Difluoro-2-phenyl-1H-indol-3-yl)-1-oxobutyl]-L-argininemethylestertrifluoroacetate;N2-[4-(5,7-DIFLUORO-2-PHENYL-1H-INDOL-3-YL)-1-OXOBUTYL]-L-ARGININE METHYL ESTER TRIFLUOROACETATE;L-803087
SMILES:	NC(NCCCC(C(OC)=O)NC(CCCC1=C(C2=CC=CC=C2)NC2=C(C=C(C=C12)F)F)=O)=N.OC(C(F)(F)F)=O
Formula:	C₂₅H₂₉F₂N₅O₃
M.Wt:	599.55000
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Cat. No.	Product name	Field of application
DC46145	Paltusotine	Paltusotine (CRN00808) is an orally active, nonpeptide selective somatostatin type 2 (SST2) receptor agonist. Paltusotine has the potential for maintaining GH and IGF-1 levels after depot somatostatin receptor ligand therapy.
DC28234	L-803087	L-803087 is a potent and selective somatostatin sst4 receptor agonist with a Ki of 0.7 nM, which is > 280-fold higher than other somatostatin receptors. L-803087 facilitates AMPA-mediated hippocampal synaptic responses in vitro and increases kainate-induced seizures in mice.